SCHEMBL23536729

SCHEMBL23536729

Cc1cc(C#N)cc(CCN)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.46
CYP2A6 P11509 2/20 0.42
CYP1A2 P05177 1/20 0.42
NOS1 P29475 2/20 0.42
NOS3 P29474 1/20 0.42
NOS2 P35228 3/20 0.37
BACE1 P56817 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ADRA2C P18825 1/20 0.35
XDH P47989 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17277608 0.87 NOS1 (0.45) TAAR1NOS1NOS3NOS2LOXL2
SCHEMBL7896912 0.84 LOXL2 (0.48) CYP2A6NOS1NOS3NOS2LOXL2
SCHEMBL16958451 0.82 NOS1 (0.40) CYP2A6NOS1NOS3NOS2ALDH1A1
SCHEMBL7358317 0.81 NOS1 (0.39) CYP2A6NOS1NOS3NOS2BACE1
SCHEMBL27748133 0.81 NOS1 (0.39) CYP2A6NOS1NOS3NOS2ALDH1A1
SCHEMBL7358314 0.81 NOS1 (0.39) CYP2A6NOS1NOS3NOS2ALDH1A1
SCHEMBL537203 0.79 TAAR1 (0.60) TAAR1CYP2A6CYP1A2NOS1NOS3
SCHEMBL3849051 0.79 TAAR1 (0.60) TAAR1CYP2A6CYP1A2NOS1NOS3
SCHEMBL22477339 0.78 CYP2A6 (0.39) CYP2A6NOS1NOS3NOS2LOXL2
SCHEMBL11982666 0.78 CYP2A6 (0.50) CYP2A6NOS1NOS3NOS2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076418-A1 SOS1 INHIBITORS Mirati Therapeutics, Inc. (US) 2022-10-26 EP disclosed
WO-2021127429-A1 SOS1 INHIBITORS Mirati Therapeutics, Inc. (US) 2021-06-24 WO disclosed