SCHEMBL23547291

SCHEMBL23547291

COC1CN(c2nc(C)n3ncc(C(C)C)c3n2)C1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 9/20 0.35
CDK2 P24941 9/20 0.35
PDE2A O00408 6/20 0.33
CDK7 P50613 2/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
CDK4 P11802 1/20 0.32
CCNE1 P24864 2/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26973961 0.78 ALDH1A1 (0.40) CDK9CDK2CCNE1
SCHEMBL26973963 0.77 CDK2 (0.37) CDK9CDK2CCNE1GSK3B
SCHEMBL26973993 0.71 CDK2 (0.33) CDK9CDK2CDK7CCNHMNAT1
SCHEMBL15245996 0.64 CDK2 (0.40) CDK9CDK2CDK7CCNHMNAT1
SCHEMBL23547295 0.64 CCNE1 (0.41) CDK2CCNE1
SCHEMBL21486451 0.64 HRH3 (0.37) CDK9CDK2CDK7CCNHMNAT1
SCHEMBL18430319 0.63 ACACB (0.45) PDE2AKCNQ3KCNQ2
SCHEMBL21481492 0.62 PTPN11 (0.38) CDK9CDK2CDK7CCNHMNAT1
SCHEMBL21481494 0.62 CDK2 (0.37) CDK9CDK2CDK7CCNHMNAT1
SCHEMBL20971704 0.61 MAPT (0.54) CDK9CDK2CDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021121390-A1 HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, INTERMEDIATE THEREOF AND APPLICATION THEREOF 苏州信诺维医药科技股份有限公司 2021-06-24 WO disclosed