SCHEMBL23547485

SCHEMBL23547485

Cc1nc(NC2CCN(C(=O)OC(C)(C)C)CC2)n2ncc(C(C)C)c2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
NPC1 O15118 1/20 0.52
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.52
HTT P42858 1/20 0.52
RAB9A P51151 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
CDK9 P50750 4/20 0.47
CDK4 P11802 1/20 0.47
CDK7 P50613 1/20 0.47
CDK2 P24941 4/20 0.41
GPR119 Q8TDV5 2/20 0.41
ADORA2A P29274 1/20 0.41
JAK1 P23458 1/20 0.41
CNR1 P21554 2/20 0.40
CCNA2 P20248 1/20 0.40
NSD2 O96028 1/20 0.40
EPHX1 P07099 1/20 0.40
IDH1 O75874 1/20 0.40
IDH2 P48735 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23529883 0.94 CDK9 (0.54) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL31064099 0.90 CDK9 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547353 0.89 ALDH1A1 (0.51) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL31064055 0.89 ALDH1A1 (0.42) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547464 0.88 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547341 0.88 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547374 0.88 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547337 0.87 ALDH1A1 (0.48) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL31063997 0.87 CDK9 (0.41) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547517 0.86 CDK9 (0.45) CDK9CDK4CDK7CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175024-A1 NEW FUSED HETEROCYCLIC COMPOUND AS CDKS INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2024-08-29 WO disclosed
CN-113004285-B Heterocyclic compound, pharmaceutical composition, preparation method, intermediate and application thereof 苏州信诺维医药科技股份有限公司 2024-05-14 CN disclosed
WO-2021121390-A1 HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, INTERMEDIATE THEREOF AND APPLICATION THEREOF 苏州信诺维医药科技股份有限公司 2021-06-24 WO disclosed
CN-113004285-A Heterocyclic compound and pharmaceutical composition, preparation method, intermediate and application thereof 苏州信诺维医药科技股份有限公司 2021-06-22 CN disclosed