SCHEMBL23547337

SCHEMBL23547337

CC(C)c1cnn2c(NC3CCN(C(=O)OC(C)(C)C)CC3)nc(S(C)(=O)=O)nc12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
GPR119 Q8TDV5 10/20 0.46
CDK9 P50750 3/20 0.41
CDK4 P11802 1/20 0.41
CDK7 P50613 1/20 0.41
CYP3A4 P08684 1/20 0.40
CDK2 P24941 2/20 0.39
ADORA2A P29274 1/20 0.39
JAK1 P23458 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31063972 0.90 GPR119 (0.41) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL19896550 0.88 GPR119 (0.48) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547485 0.87 ALDH1A1 (0.52) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547353 0.86 ALDH1A1 (0.51) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL31064133 0.86 GPR119 (0.45) GPR119CDK9CDK2
SCHEMBL23547374 0.84 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547464 0.84 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23547341 0.84 ALDH1A1 (0.49) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL23529883 0.83 CDK9 (0.54) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL19896539 0.83 USP30 (0.45) ALDH1A1NPC1MAPTMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175024-A1 NEW FUSED HETEROCYCLIC COMPOUND AS CDKS INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2024-08-29 WO disclosed
CN-117843642-A Difunctional compound and application thereof 麦科萨药业(苏州)有限公司 2024-04-09 CN disclosed
WO-2021121390-A1 HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, INTERMEDIATE THEREOF AND APPLICATION THEREOF 苏州信诺维医药科技股份有限公司 2021-06-24 WO disclosed