SCHEMBL2354773

SCHEMBL2354773

O=C(OCc1ccccc1)N1CCN(c2cccc3[nH]ccc23)CC1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GOT1 P17174 13/20 0.60
DRD2 P14416 1/20 0.60
DRD4 P21917 1/20 0.60
DRD3 P35462 1/20 0.60
GAA P10253 3/20 0.56
MAPT P10636 2/20 0.56
RECQL P46063 1/20 0.55
TMEM97 Q5BJF2 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
MAPK14 Q16539 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228008 0.80 GOT1 (0.70) GOT1DRD2DRD4DRD3GAA
SCHEMBL31134492 0.80 ALDH1A1 (0.51) GAAMAPTTMEM97SIGMAR1MEN1
SCHEMBL2228656 0.80 DRD2 (0.45) DRD2DRD4DRD3TMEM97SIGMAR1
SCHEMBL1537795 0.79 GAA (0.60) GOT1GAAMAPTRECQL
SCHEMBL30885791 0.79 GAA (0.60) GOT1GAAMAPTRECQL
SCHEMBL2229131 0.78 TMEM97 (0.47) GAAMAPTTMEM97SIGMAR1MEN1
SCHEMBL31414573 0.78 TMEM97 (0.47) GAAMAPTTMEM97SIGMAR1MEN1
SCHEMBL5362589 0.78 SMN1; SMN2 (0.72) GAAMAPTTMEM97SIGMAR1MEN1
SCHEMBL31414524 0.77 TMEM97 (0.46) DRD2DRD3GAAMAPTTMEM97
SCHEMBL3970912 0.77 MEN1 (0.76) GAAMEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed
WO-2011088836-A1 NOVEL 4-(ARYL-4-SULFONYL)-6,6a,7,8,9,10-HEXAHYDRO-4H-4,8,10a-TRIAZA-ACEPHENANTHRYLENE AND 3-ARYLSULFONYL-6,6a,7,8,9,10-HEXAHYDRO-3H-3,8,10a-TRIAZA-CYCLOPENTA[C]FLUORENE DERIVATIVES AS SEROTONIN 5-HT6 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed