SCHEMBL2357417

SCHEMBL2357417

CCNc1ncnc2c(C(=O)Nc3cc(NCc4cc(-n5cnc(C)c5)cc(C(F)(F)F)c4)ccc3C)csc12

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.47
BCR P11274 3/20 0.47
CSF1R P07333 1/20 0.47
EPHB2 P29323 1/20 0.47
RAF1 P04049 1/20 0.44
HCK P08631 1/20 0.44
NR2C2 P49116 1/20 0.44
BTK Q06187 1/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44
BRAF P15056 4/20 0.43
MAPT P10636 1/20 0.43
NR2E1 Q9Y466 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359007 0.94 CSF1R (0.47) ABL1BCRCSF1REPHB2RAF1
SCHEMBL2357420 0.91 ABL1 (0.51) ABL1BCRCSF1REPHB2RAF1
SCHEMBL12433883 0.90 CSF1R (0.59) ABL1BCRCSF1REPHB2RAF1
SCHEMBL2358401 0.88 BRAF (0.46) ABL1BCRCSF1REPHB2RAF1
SCHEMBL2359059 0.86 EPHB2 (0.50) ABL1BCRCSF1REPHB2RAF1
SCHEMBL2365076 0.85 KDM4E (0.44) ABL1BCRCSF1REPHB2RAF1
SCHEMBL2359009 0.83 EPHB2 (0.53) ABL1BCRCSF1REPHB2RAF1
SCHEMBL12433483 0.82 CSF1R (0.62) ABL1BCRCSF1REPHB2RAF1
SCHEMBL19057073 0.82 ABL1 (0.49) ABL1BCRRAF1BRAFNR2E1
SCHEMBL14717868 0.81 CSF1R (0.59) ABL1BCRCSF1REPHB2RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed