SCHEMBL2359604

SCHEMBL2359604

O=C(O)N1Cc2ccccc2-n2cnnc2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.40
NOTUM Q6P988 2/20 0.40
RIPK1 Q13546 5/20 0.35
CYP11B2 P19099 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
OPRK1 P41145 1/20 0.34
PDE4D Q08499 1/20 0.34
GAPDH P04406 1/20 0.34
CASP6 P55212 1/20 0.33
CYP11B1 P15538 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RYR2 Q92736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474337 0.81 MAPK1 (0.46) NAMPTNOTUM
SCHEMBL1388134 0.78 KDM4E (0.43) NOTUMRIPK1ALDH1A1HDAC8
SCHEMBL16207990 0.77 TSHR (0.38) NAMPTNOTUMRIPK1ALDH1A1CACNA1G
SCHEMBL9851802 0.73 CYP11B2 (0.41) NOTUMRIPK1CYP11B2ALDH1A1OPRK1
SCHEMBL29758685 0.72 NOTUM (0.64) NAMPTNOTUMHSP90AA1HSP90AB1NPC1
SCHEMBL2533362 0.72 NOTUM (0.64) NAMPTNOTUMHSP90AA1HSP90AB1NPC1
SCHEMBL11778334 0.72 CYP11B2 (0.54) RIPK1CYP11B2ALDH1A1OPRK1PDE4D
SCHEMBL29500932 0.70 CYP1A2 (0.44) NOTUMRIPK1CYP11B2ALDH1A1OPRK1
SCHEMBL21061364 0.69 CYP11B2 (0.45) NOTUMCYP11B2ALDH1A1OPRK1PDE4D
SCHEMBL29500960 0.69 CYP11B2 (0.36) NOTUMRIPK1CYP11B2ALDH1A1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356123-A1 SPIRO-5,6-DIHYDRO-4H-2,3,5,10B-TETRAAZA-BENZO[E]AZULENES F. Hoffmann-La Roche AG (CH) 2011-08-17 EP claimed