SCHEMBL9851802

SCHEMBL9851802

c1ccc2c(c1)Cc1nncn1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.41
OPRK1 P41145 1/20 0.38
PDE4D Q08499 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP11B1 P15538 2/20 0.35
HPGD P15428 1/20 0.34
AADAT Q8N5Z0 1/20 0.34
NOTUM Q6P988 1/20 0.33
RIPK1 Q13546 3/20 0.32
GABRA1 P14867 2/20 0.31
GABRA2 P47869 2/20 0.31
GABRB2 P47870 2/20 0.31
SLC22A2 O15244 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
DRD1 P21728 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29500932 0.88 CYP1A2 (0.44) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL11778334 0.83 CYP11B2 (0.54) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL21061364 0.80 CYP11B2 (0.45) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL2340498 0.79 AVPR1A (0.38) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL5278269 0.79 AVPR1A (0.38) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
Hydrochloric Acid SCHEMBL5277480 0.78 AVPR1A (0.38) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL29500960 0.76 CYP11B2 (0.36) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL21061622 0.76 AADAT (0.40) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL29848695 0.73 AVPR1A (0.43) CYP11B2OPRK1PDE4DALDH1A1CYP11B1
SCHEMBL2359604 0.73 NAMPT (0.40) CYP11B2OPRK1PDE4DALDH1A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0406719-A1 4h-indolo(1,2-d)(1,2,4)triazolo (4,3-a)(1,4)benzodiazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed