SCHEMBL2361917

SCHEMBL2361917

COc1cc(CN2C(=O)CC[C@@H]2CO)c(-c2ccc[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.36
HCRTR1 O43613 13/20 0.36
CYP3A4 P08684 3/20 0.36
PDK2 Q15119 1/20 0.35
GYS1 P13807 1/20 0.31
F2 P00734 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361921 1.00 HCRTR2 (0.36) HCRTR2HCRTR1CYP3A4PDK2GYS1
SCHEMBL11888716 1.00 HCRTR2 (0.36) HCRTR2HCRTR1CYP3A4PDK2GYS1
SCHEMBL2354400 0.87 GYS1 (0.41) HCRTR2HCRTR1CYP3A4GYS1F2
SCHEMBL2364358 0.87 GYS1 (0.41) HCRTR2HCRTR1CYP3A4GYS1F2
SCHEMBL2364234 0.84 ADRA1A (0.37) HCRTR2HCRTR1CYP3A4GYS1
SCHEMBL2364233 0.84 ADRA1A (0.37) HCRTR2HCRTR1CYP3A4GYS1
SCHEMBL3314212 0.81 CYP3A4 (0.40) CYP3A4
SCHEMBL2363467 0.80 CYP3A4 (0.43) CYP3A4
SCHEMBL2353888 0.78 ACHE (0.41) CYP3A4
SCHEMBL2347996 0.78 HCRTR1 (0.38) HCRTR2HCRTR1PDK2GYS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8232271-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2012-07-31 US claimed
EP-2350007-A1 HETEROCYCLIC ANTIVIRAL ARYLPYRIDONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-08-03 EP claimed
WO-2010049331-A1 HETEROCYCLIC ANTIVIRAL ARYLPYRIDONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-05-06 WO claimed