SCHEMBL2362098

SCHEMBL2362098

COC(=O)c1ccc2c(c1)nc(C(Cl)(Cl)Cl)n2C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
LMNA P02545 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
MAPT P10636 1/20 0.50
FGFR1 P11362 1/20 0.48
EHMT2 Q96KQ7 1/20 0.45
PTGER4 P35408 2/20 0.44
ACSS2 Q9NR19 2/20 0.44
HDAC6 Q9UBN7 3/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
CNR2 P34972 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
ITK Q08881 1/20 0.42
HTT P42858 2/20 0.42
ALOX15 P16050 1/20 0.42
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10238325 0.86 KDM4E (0.52) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL3370266 0.85 HCAR3 (0.50) KDM4ENPC1RAB9AFGFR1PTGER4
SCHEMBL2362614 0.84 KDM4E (0.56) KDM4EEHMT2PTGER4ACSS2CNR2
SCHEMBL19029395 0.82 KDM4E (0.56) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL31489 0.80 RAB9A (0.72) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL29989068 0.80 RAB9A (0.72) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL9412502 0.80 KMT2A (0.44) LMNANPC1RAB9AMAPTPTGER4
SCHEMBL28439988 0.79 KDM4E (0.56) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL30897550 0.79 KDM4E (0.56) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL4259457 0.79 KDM4E (0.56) KDM4ELMNANPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed