SCHEMBL2362210

SCHEMBL2362210

CS(=O)(=O)c1ccc(O[C@@H](F)C(C#CCF)NCC(CS(=O)(=O)Cc2cccnc2)C(=O)NC2(C#N)CC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.37
CTSS P25774 13/20 0.36
CTSL P07711 12/20 0.36
CTSB P07858 8/20 0.36
CTSV O60911 1/20 0.34
CTSF Q9UBX1 1/20 0.34
NAMPT P43490 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062859 0.82 CTSS (0.40) CTSKCTSSCTSLCTSBCTSV
SCHEMBL15062861 0.82 CTSS (0.40) CTSKCTSSCTSLCTSBCTSV
SCHEMBL2362018 0.75 CTSS (0.45) CTSKCTSSCTSLCTSBCTSV
SCHEMBL15062851 0.70 CTSS (0.40) CTSKCTSSCTSLCTSBCTSV
SCHEMBL15062850 0.70 CTSS (0.40) CTSKCTSSCTSLCTSBCTSV
SCHEMBL15062892 0.67 CTSS (0.54) CTSKCTSSCTSLCTSB
SCHEMBL2346448 0.67 CTSS (0.54) CTSKCTSSCTSLCTSB
SCHEMBL2342699 0.67 MMP1 (0.41) CTSKCTSSCTSLCTSB
SCHEMBL15062802 0.66 NAMPT (0.35) CTSSCTSLCTSBNAMPT
SCHEMBL15062801 0.66 NAMPT (0.35) CTSSCTSLCTSBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Virobay, Inc. (US) 2011-08-31 EP claimed
WO-2010056877-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY, INC. (US) 2010-05-20 WO claimed