SCHEMBL15062859

SCHEMBL15062859

CC#C[C@H](NC[C@@H](CS(=O)(=O)Cc1cccnc1)C(=O)NC1(C#N)CC1)C(F)(F)Oc1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.40
CTSL P07711 11/20 0.40
CTSK P43235 10/20 0.40
CTSB P07858 8/20 0.40
CTSV O60911 1/20 0.38
CTSF Q9UBX1 1/20 0.38
NAMPT P43490 1/20 0.35
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
MMP14 P50281 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062861 1.00 CTSS (0.40) CTSSCTSLCTSKCTSBCTSV
SCHEMBL15062851 0.88 CTSS (0.40) CTSSCTSLCTSKCTSBCTSV
SCHEMBL15062850 0.88 CTSS (0.40) CTSSCTSLCTSKCTSBCTSV
SCHEMBL2362018 0.84 CTSS (0.45) CTSSCTSLCTSKCTSBCTSV
SCHEMBL2362210 0.82 CTSK (0.37) CTSSCTSLCTSKCTSBCTSV
SCHEMBL15062802 0.81 NAMPT (0.35) CTSSCTSLCTSBNAMPTMMP1
SCHEMBL15062801 0.81 NAMPT (0.35) CTSSCTSLCTSBNAMPTMMP1
SCHEMBL15062930 0.79 CTSL (0.38) CTSSCTSLCTSKCTSBMMP1
SCHEMBL15062929 0.79 CTSL (0.38) CTSSCTSLCTSKCTSBMMP1
SCHEMBL15062923 0.77 CTSS (0.45) CTSSCTSLCTSKCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP claimed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP claimed
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP disclosed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP disclosed