SCHEMBL2362289

SCHEMBL2362289

CC(C)(C)c1c(C=O)ccc2[nH]cnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.34
PARP1 P09874 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
PDE2A O00408 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
POLB P06746 1/20 0.33
EGFR P00533 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
MMP12 P39900 1/20 0.33
HDAC1 Q13547 1/20 0.32
CYP3A4 P08684 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24241002 0.78 MEN1 (0.37) LMNAPARP1ALDH1A1PKMMEN1
SCHEMBL17307154 0.76 DPP4 (0.40) LMNAPARP1ALDH1A1PKMPDE2A
SCHEMBL6364767 0.76 LMNA (0.38) LMNAPARP1ALDH1A1PKMPDE2A
SCHEMBL18405893 0.76 LMNA (0.38) LMNAPARP1ALDH1A1PKMPDE2A
SCHEMBL24854117 0.75 LMNA (0.37) LMNAPARP1ALDH1A1PKMPDE2A
SCHEMBL22380086 0.71 ALDH1A1 (0.40) LMNAPARP1ALDH1A1PKMPDE2A
SCHEMBL2339392 0.71 LMNA (0.32) LMNAPARP1MEN1KMT2ACCR1
SCHEMBL534330 0.70 PARP1 (0.50) LMNAPARP1ALDH1A1MEN1KMT2A
SCHEMBL6397525 0.67 LMNA (0.42) LMNAPARP1ALDH1A1PKMMEN1
SCHEMBL4246899 0.65 PDPK1 (0.39) LMNAPARP1ALDH1A1PKMPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed