SCHEMBL23628709

SCHEMBL23628709

CCC(CO)NC(=O)c1ccc(OC)nc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 6/20 0.56
GABRA1 P14867 5/20 0.55
NNMT P40261 1/20 0.50
NR1I2 O75469 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2C9 P11712 1/20 0.46
IDO1 P14902 1/20 0.46
CYP2C19 P33261 1/20 0.46
KCNH2 Q12809 1/20 0.46
HTT P42858 1/20 0.46
FYN P06241 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
GRN P28799 1/20 0.45
SORT1 Q99523 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL702548 0.85 TAS1R3 (0.63) GABRA1NNMTTAS1R3TAS1R1GRN
SCHEMBL3436035 0.81 GRN (0.50) GABRA5GABRA1NNMTTAS1R3TAS1R1
SCHEMBL20812214 0.81 NNMT (0.60) GABRA5GABRA1NNMTGRNSORT1
SCHEMBL13403407 0.81 HDAC6 (0.54) GABRA5GABRA1NNMTHTTTAS1R3
SCHEMBL5784282 0.78 NNMT (0.50) GABRA5GABRA1NNMTNR1I2CYP2C8
SCHEMBL23628710 0.78 NNMT (0.50) GABRA5GABRA1NNMTTAS1R3TAS1R1
SCHEMBL1882423 0.76 NNMT (0.67) GABRA1NNMTHTTHDAC6
SCHEMBL24247501 0.76 GABRA1 (0.55) GABRA5GABRA1TAS1R3TAS1R1
SCHEMBL14516103 0.75 NNMT (0.64) GABRA5NNMTHTTHDAC6
SCHEMBL5784288 0.74 GRN (0.44) GABRA5GABRA1NNMTNR1I2CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3847154-A1 CARBOXAMIDE AND SULFONAMIDE DERIVATIVES USEFUL AS TEAD MODULATORS F. Hoffmann-La Roche AG (CH) 2021-07-14 EP disclosed