SCHEMBL2364574

SCHEMBL2364574

CC(c1ccccc1)c1cnc(-c2cnn3ccncc23)nc1N

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
DYRK1A Q13627 1/20 0.33
ADORA2A P29274 3/20 0.32
ADORA1 P30542 3/20 0.32
JAK2 O60674 2/20 0.32
EPHB3 P54753 1/20 0.31
ROCK2 O75116 1/20 0.30
USP1 O94782 1/20 0.30
LDHA P00338 1/20 0.30
LDHB P07195 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230884 0.87 JAK2 (0.42) PIK3CDPIK3R1PIK3CAPIK3CBPIK3CG
SCHEMBL2233315 0.75 JAK2 (0.52) JAK2JAK3
Toluene SCHEMBL2342437 0.74 DYRK1A (0.37) DYRK1AEPHB3
SCHEMBL1693166 0.72 USP1 (0.63) JAK2USP1JAK3
SCHEMBL2347275 0.69 EPHB3 (0.39) DYRK1AEPHB3
SCHEMBL4382927 0.68 P2RX3 (0.49) PIK3CA
SCHEMBL3962873 0.68 P2RX3 (0.49) PIK3CA
SCHEMBL2233691 0.67 MAPT (0.36) DYRK1AEPHB3
SCHEMBL2230590 0.67 DYRK1A (0.35) DYRK1AEPHB3
SCHEMBL2231287 0.66 ACVR2A (0.39) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101161-A1 PYRAZOLE DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2011-08-25 WO disclosed