SCHEMBL23652014

SCHEMBL23652014

CCOc1ccnc2cc(OCc3ccccc3)ccc12

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
GRM4 Q14833 2/20 0.51
MAOA P21397 1/20 0.48
TLR8 Q9NR97 1/20 0.47
DYRK1A Q13627 1/20 0.46
ALOX5 P09917 1/20 0.45
APP P05067 1/20 0.45
MET P08581 5/20 0.44
PRKACG P22612 1/20 0.44
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19968424 0.89 CYP3A4 (0.57) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL2329005 0.86 CYP3A4 (0.55) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL24411225 0.86 CYP3A4 (0.55) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL29214652 0.84 CYP3A4 (0.52) CYP3A4GRM4MAOATLR8ALOX5
SCHEMBL28665368 0.83 CYP3A4 (0.51) CYP3A4GRM4MAOB
SCHEMBL29214660 0.83 CYP3A4 (0.51) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL13443841 0.80 HTR1A (0.57) CYP3A4APPMETPRKACG
SCHEMBL3898712 0.79 CYP3A4 (0.58) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL311094 0.79 CYP3A4 (0.58) CYP3A4GRM4MAOATLR8DYRK1A
SCHEMBL30153587 0.79 CYP3A4 (0.58) CYP3A4GRM4MAOATLR8DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3510036-B1 IMIDAZOQUINOLINE DERIVATIVES AND THEIR USE IN THERAPY GLAXOSMITHKLINE BIOLOGICALS SA (BE) 2021-07-21 EP disclosed