SCHEMBL28665368

SCHEMBL28665368

O=C(O)COc1ccnc2cc(OCc3ccccc3)ccc12

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
GRM4 Q14833 1/20 0.48
PPARD Q03181 3/20 0.48
PPARG P37231 2/20 0.48
FFAR1 O14842 5/20 0.47
PLAU P00749 1/20 0.46
PLAT P00750 1/20 0.46
MAOB P27338 1/20 0.44
NR4A2 P43354 2/20 0.44
FFAR4 Q5NUL3 1/20 0.44
P2RY14 Q15391 1/20 0.44
PTPN7 P35236 1/20 0.43
NR4A1 P22736 1/20 0.43
NR4A3 Q92570 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29214652 0.84 CYP3A4 (0.52) CYP3A4GRM4PLAUPLATMAOB
SCHEMBL24411225 0.83 CYP3A4 (0.55) CYP3A4GRM4PLAUPLATMAOB
SCHEMBL2329005 0.83 CYP3A4 (0.55) CYP3A4GRM4PLAUPLATMAOB
SCHEMBL23652014 0.83 CYP3A4 (0.55) CYP3A4GRM4MAOB
SCHEMBL19968424 0.83 CYP3A4 (0.57) CYP3A4GRM4MAOB
SCHEMBL2700581 0.82 MET (0.54) CYP3A4
SCHEMBL29878429 0.82 MET (0.54) CYP3A4
SCHEMBL4299513 0.80 KDM4E (0.43)
SCHEMBL311094 0.79 CYP3A4 (0.58) CYP3A4GRM4PLAUPLATMAOB
SCHEMBL30153587 0.79 CYP3A4 (0.58) CYP3A4GRM4PLAUPLATMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113788835-B Triazole tetrazine compound containing morpholine and quinoline ring and preparation method and application thereof 台州职业技术学院 2022-08-26 CN disclosed
CN-113788835-A Triazole tetrazine compound containing morpholine and quinoline ring and preparation method and application thereof 台州职业技术学院 2021-12-14 CN disclosed