SCHEMBL2365245

SCHEMBL2365245

COc1cccc(CN2CC3CNCC(C2)O3)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.55
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 3/20 0.52
GAA P10253 1/20 0.47
CMA1 P23946 1/20 0.47
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
DRD2 P14416 2/20 0.46
HTR1A P08908 1/20 0.46
HTR2B P41595 1/20 0.46
MAPT P10636 1/20 0.46
EED O75530 1/20 0.45
LPO P22079 1/20 0.45
DRD3 P35462 1/20 0.45
FAAH O00519 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1618174 0.78 FUCA1 (0.50) SIGMAR1ALDH1A1DRD2DRD3
SCHEMBL2330991 0.78 ADRB1 (0.55) KDM4EALDH1A1DRD2MAPTMEN1
SCHEMBL2921693 0.77 SIGMAR1 (0.63) SIGMAR1KDM4EALDH1A1GAACMA1
SCHEMBL2918653 0.77 SIGMAR1 (0.63) SIGMAR1KDM4EALDH1A1GAACMA1
Hydrochloric Acid SCHEMBL1619305 0.77 FUCA1 (0.49) SIGMAR1ALDH1A1DRD2DRD3
SCHEMBL2910904 0.76 SIGMAR1 (0.57) SIGMAR1KDM4EALDH1A1GAACMA1
SCHEMBL28186295 0.75 SIGMAR1 (0.90) SIGMAR1KDM4EALDH1A1GAALMNA
SCHEMBL20804357 0.75 SIGMAR1 (0.90) SIGMAR1KDM4EALDH1A1GAALMNA
SCHEMBL3847058 0.75 SIGMAR1 (0.72) SIGMAR1KDM4EALDH1A1GAADRD2
SCHEMBL29463795 0.75 SIGMAR1 (0.72) SIGMAR1KDM4EALDH1A1GAADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356125-A1 DERIVATIVES OF OXABISPIDINE AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS Targacept, Inc. (US) 2011-08-17 EP disclosed
WO-2010002971-A1 DERIVATIVES OF OXABISPIDINE AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-01-07 WO disclosed