SCHEMBL23660879

SCHEMBL23660879

COC(=O)c1cc(F)c2c(c1Br)OCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 7/20 0.41
TARBP2 Q15633 2/20 0.38
SOS1 Q07889 1/20 0.37
PKM P14618 2/20 0.36
GAA P10253 3/20 0.34
MAPK1 P28482 3/20 0.34
ALOX15 P16050 2/20 0.34
HPGD P15428 4/20 0.34
ATM Q13315 1/20 0.34
MAPK10 P53779 1/20 0.34
HIF1A Q16665 1/20 0.34
SMN1; SMN2 Q16637 5/20 0.33
CASP1 P29466 2/20 0.33
CASP7 P55210 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
POLB P06746 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23660880 0.83 ALDH1A1 (0.42) KDM4EALDH1A1TARBP2PKMGAA
SCHEMBL5360890 0.82 KDM4E (0.45) KDM4EALDH1A1TARBP2PKMGAA
SCHEMBL23660877 0.81 SMN1; SMN2 (0.40) KDM4EALDH1A1GAAMAPK1HPGD
SCHEMBL30184719 0.80 KDM4E (0.45) KDM4EALDH1A1SOS1PKMHPGD
SCHEMBL25045981 0.80 KDM4E (0.45) KDM4EALDH1A1SOS1PKMHPGD
SCHEMBL9716376 0.76 KDM4E (0.48) KDM4EALDH1A1GAAMAPK1HPGD
SCHEMBL30507860 0.76 KDM4E (0.41) KDM4EALDH1A1TARBP2SOS1PKM
SCHEMBL29054615 0.76 KDM4E (0.48) KDM4EALDH1A1TARBP2PKMGAA
SCHEMBL29054666 0.76 KDM4E (0.41) KDM4EALDH1A1TARBP2SOS1PKM
SCHEMBL17714988 0.75 TARBP2 (0.48) KDM4EALDH1A1TARBP2PKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021143822-A1 BICYCLIC IMIDE DERIVATIVE, PREPARATION METHOD THEREOF, AND APPLICATION THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2021-07-22 WO disclosed