SCHEMBL23664151

SCHEMBL23664151

Cc1cnc(N2CCOCC2)c(-c2cccc(S(C)(=O)=O)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.54
PIK3CG P48736 1/20 0.54
MTOR P42345 3/20 0.53
PIK3CB P42338 2/20 0.52
JAK2 O60674 3/20 0.47
JAK3 P52333 3/20 0.47
ATR Q13535 3/20 0.47
ATRIP Q8WXE1 2/20 0.47
RAF1 P04049 4/20 0.47
BRAF P15056 4/20 0.47
PTK2 Q05397 2/20 0.46
LRRK2 Q5S007 2/20 0.45
STK4 Q13043 1/20 0.45
STK3 Q13188 1/20 0.45
ACVR1 Q04771 2/20 0.45
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170360 0.85 PIK3CA (0.51) PIK3CAPIK3CGMTORPIK3CBJAK2
SCHEMBL31301537 0.76 LRRK2 (0.72) LRRK2STK4STK3
SCHEMBL6169775 0.76 CNR2 (0.44) PIK3CAPIK3CGMTORJAK2LRRK2
SCHEMBL6169601 0.74 PTGS2 (0.58) KDM4EATM
SCHEMBL6069405 0.74 PTGS2 (0.48) JAK2LRRK2ACVR1
SCHEMBL6069433 0.74 RIPK2 (0.50) PIK3CAJAK2ATRPTK2STK3
SCHEMBL6169315 0.73 PTGS2 (0.57) KDM4EATM
SCHEMBL5204774 0.73 PTGS2 (0.60) JAK2JAK3ATRLRRK2KMT2A
SCHEMBL6170358 0.72 PTGS2 (0.63) PIK3CAPIK3CG
SCHEMBL6170721 0.72 PTGS2 (0.51) PIK3CAMTORPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021143927-A1 COMPOUND ACTING AS BCR-ABL INHIBITOR 正大天晴药业集团股份有限公司 2021-07-22 WO disclosed