SCHEMBL2369286

SCHEMBL2369286

CCOC(=O)C(C(=O)OCC)c1nc(NCc2cccc(C)n2)c2c(-c3ccc(F)cc3)csc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 1/20 0.37
PTPN1 P18031 1/20 0.36
ESR1 P03372 3/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
LMNA P02545 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 1/20 0.35
TNF P01375 1/20 0.35
MAPK1 P28482 1/20 0.35
NOD1 Q9Y239 1/20 0.35
SLC26A6 Q9BXS9 3/20 0.35
SCN9A Q15858 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3415878 0.92 ESR1 (0.44) ESR1ALDH1A1LMNARXFP1KDM4E
Butane SCHEMBL6359950 0.90 ESR1 (0.38) ESR1ALDH1A1HPGDLMNARXFP1
SCHEMBL3386697 0.89 TNF (0.48) PTPN1ESR1MAPTALDH1A1KDM4E
SCHEMBL2369294 0.88 TGM2 (0.36) PTPN1ESR1MAPTALDH1A1HPGD
SCHEMBL2368960 0.86 ESR1 (0.39) ESR1ALDH1A1HPGDLMNARXFP1
SCHEMBL3383460 0.85 PRKCZ (0.43) PRKCZMAPTALDH1A1HPGDLMNA
SCHEMBL3384941 0.85 ALDH1A1 (0.38) MAPTALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL2369471 0.85 ALDH1A1 (0.47) PRKCZESR1MAPTALDH1A1HPGD
SCHEMBL2368543 0.82 TNF (0.56) ESR1ALDH1A1LMNASMN1; SMN2TNF
SCHEMBL3415890 0.80 ESR1 (0.40) ESR1ALDH1A1LMNASMN1; SMN2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022076-B2 Thieno[2,3-d]pyrimidine derivatives as potassium channel modulators; antiarrhythmia agents XENTION LIMITED (GB) 2011-09-20 US disclosed
EP-1641803-B3 THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS XENTION LTD (GB) 2010-12-08 EP disclosed
EP-1641803-B1 THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS XENTION LTD (GB) 2009-03-18 EP disclosed