SCHEMBL2369340

SCHEMBL2369340

O=CC(Cc1ccccc1)NC(=O)O

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 8/20 0.61
ACE P12821 1/20 0.56
CTSB P07858 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865652 1.00 CAPN1 (0.61) CAPN1ACECTSB
SCHEMBL3292711 1.00 CAPN1 (0.61) CAPN1ACECTSB
SCHEMBL16932220 0.90 CAPN1 (0.52) CAPN1ACECTSB
SCHEMBL20204724 0.87 CTSB (0.55) CAPN1ACECTSB
SCHEMBL20204721 0.87 CTSB (0.55) CAPN1ACECTSB
SCHEMBL2293365 0.86 CAPN1 (0.53) CAPN1CTSB
SCHEMBL10045690 0.86 CAPN1 (0.58) CAPN1ACECTSB
SCHEMBL2911854 0.86 CAPN1 (0.58) CAPN1ACECTSB
SCHEMBL12125815 0.86 CAPN1 (0.58) CAPN1ACECTSB
SCHEMBL2269431 0.86 CAPN1 (0.58) CAPN1ACECTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2895492-A1 PROCESS FOR PREPARING OF BORTEZOMIB Cipla Limited (IN) 2015-07-22 EP claimed
WO-2014041324-A1 PROCESS FOR PREPARING OF BORTEZAMIB CIPLA LIMITED (IN) 2014-03-20 WO claimed
EP-4373825-A1 NITRILE SUMO INHIBITORS AND USES THEREOF Suvalent Therapeutics, Inc. (US) 2024-05-29 EP disclosed
CN-117836270-A USP30 inhibitors and uses thereof 文森雷生物科学股份有限公司 2024-04-05 CN disclosed
EP-4305021-A1 USP30 INHIBITORS AND USES THEREOF Vincere Biosciences, Inc. (US) 2024-01-17 EP disclosed
EP-3788031-B1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF LANDSTEINER GENMED S L (ES) 2023-09-27 EP disclosed
WO-2023004376-A1 NITRILE SUMO INHIBITORS AND USES THEREOF Suvalent Therapeutics, Inc. (US) 2023-01-26 WO disclosed
WO-2022192562-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. (US) 2022-09-15 WO disclosed
US-20220274976-A1 COMPOSITIONS, FORMULATIONS AND METHODS FOR TREATING OCULAR DISEASES EyePoint, Inc. 2022-09-01 US disclosed
US-11242312-B2 Dipeptidyl ketoamide meta-methoxyphenyl derivatives and uses thereof LANDSTEINER GENMED, S.L. (ES) 2022-02-08 US disclosed
US-20210317075-A1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF LANDSTEINER GENMED, S.L. (ES) 2021-10-14 US disclosed
US-20100137633-A1 Process For Deacetalisation Of Alpha Aminoacetals CLARIANT SPECIALTY FINE CHEMICALS (FRANCE) (FR) 2010-06-03 US disclosed
EP-2152664-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS Brystol-Myers Squibb Company (US) 2010-02-17 EP disclosed
EP-2137139-A1 PROCESS OF DEACETALISATION OF ALPHA AMINOACETALS Clariant Specialty Fine Chemicals (France) (FR) 2009-12-30 EP disclosed
WO-2008157162-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-24 WO disclosed
WO-2008125486-A1 PROCESS OF DEACETALISATION OF ALPHA AMINOACETALS CLARIANT SPECIALTY FINE CHEMICALS (FRANCE) (FR) 2008-10-23 WO disclosed
US-5583248-A Amino acid derivatives having antiviral activity HOFFMANN-LA ROCHE INC. (US) 1996-12-10 US disclosed
US-5294720-A Viricides THE DUPONT MERCK PHARMACEUTICAL CO. (US) 1994-03-15 US disclosed
US-5135914-A Controlling hypertension, hyperaldosteronism, and congestive heart failure WARNER-LAMBERT COMPANY (US) 1992-08-04 US disclosed
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137633-A1 Process For Deacetalisation Of Alpha Aminoacetals ALDH7A1, AADAT, AASDHPPT CAPN1 1431/4885ACE 85/4885CTSB 1587/4885
US-11242312-B2 Dipeptidyl ketoamide meta-methoxyphenyl derivatives and uses thereof DPP4, DPP7, DPP3 CAPN1 25/4885ACE 9/4885CTSB 159/4885
US-20220274976-A1 COMPOSITIONS, FORMULATIONS AND METHODS FOR TREATING OCULAR DISEASES TIE1, TEK, KDR CAPN1 4685/4885ACE 1795/4885CTSB 1930/4885
US-20210317075-A1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF DPP4, DPP7, DPP3 CAPN1 25/4885ACE 9/4885CTSB 159/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.