SCHEMBL23699028

SCHEMBL23699028

COc1ccc2nc(C#N)ccc2c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.47
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42
GRM5 P41594 2/20 0.39
KCNH2 Q12809 2/20 0.39
KDM4E B2RXH2 3/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CDK2 P24941 1/20 0.38
CLK1 P49759 1/20 0.38
AKR1B10 O60218 1/20 0.36
AKR1A1 P14550 1/20 0.36
AKR1B1 P15121 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25873382 0.81 NQO1 (0.40) NQO1ABCC8KCNJ11KDM4EMAPT
SCHEMBL16550190 0.78 NQO1 (0.50) NQO1ABCC8KCNJ11GRM5KCNH2
SCHEMBL8745729 0.78 NOTUM (0.39) NQO1ABCC8KCNJ11KDM4EPDE4A
SCHEMBL935572 0.71 PSMB8 (0.43) ABCC8KCNJ11KDM4EALDH1A1NPSR1
SCHEMBL14747557 0.71 CTSS (0.38) NQO1ABCC8KCNJ11KDM4EMAPT
SCHEMBL9575279 0.71 IMPDH2 (0.57) KDM4EMAPTALDH1A1AKR1B10AKR1A1
SCHEMBL4702849 0.69 PDE4A (0.48) NQO1KDM4EPDE4APDE4BPDE4C
SCHEMBL26931898 0.69 NQO1 (0.47) NQO1GRM5KCNH2KDM4EPDE10A
SCHEMBL7226370 0.68 NQO1 (0.47) NQO1KDM4EPDE4APDE4BPDE4C
SCHEMBL31432803 0.68 NQO1 (0.47) NQO1KDM4EPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12065422-B2 Reagents and process for direct C—H functionalization STUDIENGESELLSCHAFT KOHLE GGMBH (DE) 2024-08-20 US disclosed
US-20230227425-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION STUDIENGESELLSCHAFT KOHLE MBH (DE) 2023-07-20 US disclosed
US-20230227425-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION STUDIENGESELLSCHAFT KOHLE MBH (DE) 2023-07-20 US disclosed
US-20220002263-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION STUDIENGESELLSCHAFT KOHLE MBH (DE) 2022-01-06 US disclosed
EP-3856734-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION Studiengesellschaft Kohle mbH (DE) 2021-08-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227425-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION CFH, DOHH, CTSH NQO1 456/4885ABCC8 4836/4885KCNJ11 4526/4885
US-20220002263-A1 REAGENTS AND PROCESS FOR DIRECT C-H FUNCTIONALIZATION CFH, DOHH, CTSH NQO1 456/4885ABCC8 4836/4885KCNJ11 4526/4885
US-12065422-B2 Reagents and process for direct C—H functionalization CFH, DOHH, CTSH NQO1 544/4885ABCC8 4826/4885KCNJ11 4535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.