SCHEMBL23699089

SCHEMBL23699089

CCOC(=O)C(C)N1CC2C(C1)C2C(=O)c1ccnc2ccc(F)cc12

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 15/20 0.44
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.38
PREP P48147 1/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
GFER P55789 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23699117 0.87 IDO1 (0.49) IDO1PREPGFER
SCHEMBL23707514 0.84 IDO1 (0.49) IDO1CYP3A4
SCHEMBL23707461 0.83 IDO1 (0.55) IDO1CYP3A4
SCHEMBL23699147 0.82 IDO1 (0.43) IDO1CYP3A4
SCHEMBL22270531 0.80 IDO1 (0.48) IDO1CYP3A4
SCHEMBL28646104 0.79 MAPT (0.41) IDO1MAPTTP53POLBCYP3A4
SCHEMBL23699124 0.79 IDO1 (0.55) IDO1CYP3A4
SCHEMBL23699135 0.77 IDO1 (0.42) IDO1CYP3A4
SCHEMBL23707462 0.77 IDO1 (0.49) IDO1CYP3A4
SCHEMBL23707506 0.77 IDO1 (0.38) IDO1MAPTTP53POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210379052-A1 QUINOLINE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITORY ACTIVITY SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD. (CN) 2021-12-09 US disclosed
EP-3858813-A1 QUINOLONE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITED ACTIVITY Shenzhen Chipscreen Biosciences Co., Ltd. (CN) 2021-08-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210379052-A1 QUINOLINE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITORY ACTIVITY IDO1, IDO2, INMT IDO1 1/4885MAPT 3101/4885TP53 903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.