SCHEMBL23699376

SCHEMBL23699376

C[C@@H](c1cccc(F)c1)[C@@H](CNC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
SYK P43405 1/20 0.40
GPR119 Q8TDV5 1/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 1/20 0.39
PPARG P37231 1/20 0.39
NCOA2 Q15596 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
GPR139 Q6DWJ6 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23699379 1.00 CTSS (0.45) CTSSCTSKSYKGPR119TSHR
SCHEMBL21903152 0.86 SYK (0.48) CTSSCTSKSYK
SCHEMBL23699059 0.86 SYK (0.48) CTSSCTSKSYK
SCHEMBL23699350 0.86 CTSS (0.44) CTSSCTSKSYKGPR119TSHR
SCHEMBL23699348 0.86 CTSS (0.44) CTSSCTSKSYKGPR119TSHR
SCHEMBL23699389 0.82 CNR2 (0.44) CTSSCTSKSYKLMNAOPRM1
SCHEMBL23699392 0.82 CNR2 (0.44) CTSSCTSKSYKLMNAOPRM1
SCHEMBL14870380 0.81 CTSS (0.46) CTSSCTSKSYKGPR119TSHR
SCHEMBL4598462 0.81 CTSS (0.46) CTSSCTSKSYKGPR119TSHR
SCHEMBL11306615 0.80 CTSS (0.45) CTSSCTSKSYKGPR119TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3858439-A1 AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2021-08-04 EP disclosed
EP-3858439-A1 AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2021-08-04 EP disclosed