SCHEMBL23707488

SCHEMBL23707488

CN(c1ccnc2ccc(F)cc12)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.52
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GPR119 Q8TDV5 14/20 0.44
CYP2C9 P11712 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
TDO2 P48775 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23359754 0.86 GPR119 (0.52) MEN1KMT2AGPR119
SCHEMBL29862979 0.86 GPR119 (0.52) MEN1KMT2AGPR119
SCHEMBL23699114 0.86 IDO1 (0.43) IDO1
SCHEMBL29923819 0.82 IDO1 (0.58) IDO1GPR119CYP2C9SMN1; SMN2TDO2
SCHEMBL21034703 0.82 IDO1 (0.58) IDO1GPR119CYP2C9SMN1; SMN2TDO2
SCHEMBL23360292 0.81 GPR119 (0.49) MEN1KMT2AGPR119
SCHEMBL29862569 0.80 USP30 (0.46) MEN1KMT2AGPR119
SCHEMBL28834092 0.80 USP30 (0.46) MEN1KMT2AGPR119
SCHEMBL28834090 0.80 USP30 (0.46) MEN1KMT2AGPR119
SCHEMBL17729205 0.80 IDO1 (0.69) IDO1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210379052-A1 QUINOLINE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITORY ACTIVITY SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD. (CN) 2021-12-09 US disclosed
EP-3858813-A1 QUINOLONE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITED ACTIVITY Shenzhen Chipscreen Biosciences Co., Ltd. (CN) 2021-08-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210379052-A1 QUINOLINE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITORY ACTIVITY IDO1, IDO2, INMT IDO1 1/4885MEN1 3118/4885KMT2A 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.