SCHEMBL2371284

SCHEMBL2371284

O=C(O)c1cccc(-c2ccccc2)c1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HNF4A P41235 1/20 0.63
TSHR P16473 1/20 0.59
CLCN2 P51788 1/20 0.54
FABP3 P05413 2/20 0.53
FABP4 P15090 2/20 0.53
FABP5 Q01469 2/20 0.53
ALDH1A1 P00352 4/20 0.52
BCAT2 O15382 1/20 0.52
ALOX15 P16050 1/20 0.50
AKR1C3 P42330 1/20 0.47
AKR1C2 P52895 1/20 0.47
AKR1C1 Q04828 1/20 0.47
MYC P01106 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19923193 0.87 TSHR (0.68) HNF4ATSHRALDH1A1ALOX15MYC
SCHEMBL9712509 0.86 HNF4A (0.52) HNF4ATSHRCLCN2FABP3FABP4
SCHEMBL17965677 0.85 TSHR (0.52) HNF4ATSHRCLCN2ALDH1A1AKR1C3
SCHEMBL3927795 0.84 CLCN2 (0.54) HNF4ATSHRCLCN2FABP3FABP4
SCHEMBL7407371 0.83 HNF4A (0.73) HNF4ATSHRFABP3FABP4FABP5
SCHEMBL2574179 0.83 MAPT (0.50) HNF4ATSHRCLCN2AKR1C3AKR1C2
SCHEMBL18936558 0.83 DCLRE1B (0.49) HNF4ATSHRFABP3FABP4
SCHEMBL3169546 0.81 FOLH1 (0.53) HNF4ATSHR
SCHEMBL2744720 0.81 TSHR (0.47) HNF4ATSHRCLCN2
SCHEMBL29386013 0.81 ALDH1A1 (0.55) HNF4ATSHRCLCN2ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113321640-B Indole compound and application thereof 中国科学院广州生物医药与健康研究院 2023-06-09 CN disclosed
CN-109111427-B Indole compound and application thereof 中国科学院广州生物医药与健康研究院 2023-06-02 CN disclosed
CN-109111427-A Indole compound and application thereof, and pharmaceutical composition and application thereof 中国科学院广州生物医药与健康研究院 2019-01-01 CN disclosed
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed
EP-2635279-A2 CHEMICAL COMPOUNDS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2013-09-11 EP disclosed
WO-2012061557-A2 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-05-10 WO disclosed
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed
EP-1919479-A2 MELANOCORTIN RECEPTOR-SPECIFIC PIPERAZINE AND KETO-PIPERAZINE COMPOUNDS Palatin Technologies, Inc. (US) 2008-05-14 EP disclosed
WO-2007021991-A2 MELANOCORTIN RECEPTOR-SPECIFIC PIPERAZINE AND KETO-PIPERAZINE COMPOUNDS PALATIN TECHNOLOGIES, INC. (US) 2007-02-22 WO disclosed
EP-1389185-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-02-18 EP disclosed
WO-2002094770-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-28 WO disclosed
EP-1183284-A1 PROCESS FOR PRODUCING ETHYLENE/OLEFIN INTERPOLYMERS EASTMAN CHEMICAL COMPANY (US) 2002-03-06 EP disclosed
WO-2000075202-A1 PROCESS FOR PRODUCING ETHYLENE/OLEFIN INTERPOLYMERS EASTMAN CHEMICAL COMPANY (US) 2000-12-14 WO disclosed