SCHEMBL23715875

SCHEMBL23715875

CC(/C=C(\C)Br)=C(/N)Cc1ccc(C)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.37
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CTBP2 P56545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
AGXT P21549 2/20 0.33
MAPK8 P45983 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23716232 0.85 IDO1 (0.36) IDO1TAAR1CTBP2L3MBTL1NPC1
SCHEMBL23716093 0.83 IDO1 (0.41) IDO1CYP1A2CYP2A6TAAR1CTBP2
SCHEMBL23716075 0.78 IDO1 (0.40) IDO1TAAR1KMT2ALMNA
SCHEMBL23716188 0.74 ANO1 (0.33)
SCHEMBL23716046 0.74 IDO1 (0.38) IDO1CYP1A2CYP2A6TAAR1CTBP2
SCHEMBL23716192 0.73 BACE1 (0.31) LMNA
SCHEMBL23716318 0.72 IDO1 (0.37) IDO1CYP1A2CYP2A6TAAR1CTBP2
SCHEMBL23715945 0.70 IDO1 (0.35) IDO1CYP1A2CYP2A6TAAR1CTBP2
SCHEMBL15964777 0.67 IDO1 (0.42) IDO1CTBP2MEN1KMT2AL3MBTL1
SCHEMBL658518 0.66 CA2 (0.67) CTBP2L3MBTL1MAPK8NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed