SCHEMBL23723787

SCHEMBL23723787

C[C@H](Oc1cc(Br)cc2c1C(=O)OC2)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 2/20 0.35
CYP3A4 P08684 1/20 0.34
SLC6A9 P48067 2/20 0.33
PDE5A O76074 1/20 0.33
PDE4A P27815 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE1C Q14123 1/20 0.33
PDE3A Q14432 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RORC P51449 1/20 0.32
MAOA P21397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23723789 1.00 KDM4E (0.37) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL31496906 0.81 KDM4E (0.38) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL31496832 0.76 CYP3A4 (0.53) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL23723834 0.75 PARP10 (0.40) RORCDHODH
SCHEMBL23723784 0.75 PARP10 (0.40) RORCDHODH
SCHEMBL28900677 0.75 KDM4E (0.33) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL23723783 0.74 RORC (0.31) RORC
SCHEMBL29914938 0.73 KDM4E (0.41) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL27002518 0.73 KDM4E (0.41) KDM4EGAASMN1; SMN2LMNACYP3A4
SCHEMBL30546380 0.72 KDM4E (0.36) KDM4EGAASMN1; SMN2LMNAPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100124-A1 HETEROCYCLIC COMPOUNDS AS DIHYDROOROTATE DEHYDROGENASE INHIBITORS Janssen Biotech, Inc. (US) 2022-12-14 EP disclosed
WO-2021156787-A1 HETEROCYCLIC COMPOUNDS AS DIHYDROOROTATE DEHYDROGENASE INHIBITORS JANSSEN BIOTECH, INC. (US) 2021-08-12 WO disclosed