SCHEMBL23732010

SCHEMBL23732010

C=C(C)c1ccc(OC)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.53
TAS1R3 Q7RTX0 9/20 0.45
TAS1R1 Q7RTX1 9/20 0.45
PDE4A P27815 3/20 0.43
PDE4B Q07343 3/20 0.43
PDE4C Q08493 3/20 0.43
PDE4D Q08499 3/20 0.43
TSHR P16473 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA7 P43166 1/20 0.41
TPMT P51580 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10414443 0.86 ALOX15 (0.39) ALOX15TAS1R3TAS1R1PDE4APDE4B
SCHEMBL11611523 0.84 PDE4A (0.43) TAS1R3TAS1R1PDE4APDE4BPDE4C
SCHEMBL8296526 0.83 CYP2C9 (0.61) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL16950467 0.83 ALOX15 (0.56) ALOX15TAS1R3TAS1R1PDE4APDE4B
SCHEMBL17833298 0.82 ALOX15 (0.51) ALOX15TAS1R3TAS1R1PDE4APDE4B
SCHEMBL7644124 0.80 TAS1R3 (0.37) ALOX15TAS1R3TAS1R1PDE4APDE4B
SCHEMBL7642683 0.80 TAS1R3 (0.38) ALOX15TAS1R3TAS1R1PDE4APDE4B
SCHEMBL10336472 0.80 TUBB1 (0.50) ALOX15PDE4APDE4BPDE4CPDE4D
SCHEMBL195793 0.80 ALDH1A1 (0.56) ALOX15TAS1R3TAS1R1TSHRCYP1A2
SCHEMBL19462991 0.80 TUBB1 (0.62) ALOX15PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021154661-A1 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-08-05 WO disclosed