SCHEMBL23735498

SCHEMBL23735498

CC(F)(F)c1cc(N)c2c(c1)CCNCC2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.37
HTR2C P28335 9/20 0.34
HTR2B P41595 9/20 0.34
HTR2A P28223 7/20 0.34
ADCY6 O43306 1/20 0.32
ADCY3 O60266 1/20 0.32
ADCY9 O60503 1/20 0.32
ADCY5 O95622 1/20 0.32
ADCY8 P40145 1/20 0.32
ADCY7 P51828 1/20 0.32
ADCY2 Q08462 1/20 0.32
ADCY1 Q08828 1/20 0.32
ADCY4 Q8NFM4 1/20 0.32
DRD2 P14416 1/20 0.30
PNMT P11086 1/20 0.30
ASIC3 Q9UHC3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19684588 0.75 PNMT (0.41) HTR2CHTR2BHTR2APNMTASIC3
SCHEMBL19684606 0.73 PNMT (0.39) HTR2CHTR2BHTR2APNMTASIC3
SCHEMBL19711570 0.73 PNMT (0.39) HTR2CHTR2BHTR2APNMTASIC3
SCHEMBL22658197 0.70 KDM4E (0.30)
SCHEMBL29433292 0.70 KDM4E (0.30)
SCHEMBL19443102 0.67 PNMT (0.51) CD44HTR2CHTR2BHTR2ADRD2
SCHEMBL19684653 0.65 HRH3 (0.38) PNMT
SCHEMBL719964 0.64 ADCY6 (0.56) CD44HTR2CHTR2BHTR2AADCY6
SCHEMBL19684597 0.64 ASIC3 (0.40) HTR2CHTR2BHTR2APNMTASIC3
SCHEMBL19406903 0.64 PNMT (0.39) HTR2CHTR2BHTR2APNMTASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464249-B1 SUBSTITUTED CARBONUCLEOSIDE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER (US) 2021-08-11 EP disclosed