SCHEMBL2373934

SCHEMBL2373934

CC(C)(C)OC(=O)Cc1cccc(C(F)(F)F)n1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.43
MAOB P27338 1/20 0.42
ADORA2A P29274 1/20 0.39
ADRB1 P08588 1/20 0.39
HCRTR1 O43613 4/20 0.39
HCRTR2 O43614 4/20 0.39
ADAMTS4 O75173 1/20 0.38
MMP13 P45452 1/20 0.38
MBOAT4 Q96T53 1/20 0.38
SYK P43405 1/20 0.36
IDH1 O75874 2/20 0.35
IDH2 P48735 2/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
GRM2 Q14416 1/20 0.35
KMT2A Q03164 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31646435 0.85 P2RX7 (0.49) P2RX7MAOBADORA2AADRB1HCRTR1
SCHEMBL26046016 0.83 P2RX7 (0.49) P2RX7MAOBADORA2AADRB1HCRTR1
SCHEMBL30864787 0.82 SYK (0.47) P2RX7MAOBMBOAT4SYKKMT2A
SCHEMBL534133 0.82 SYK (0.47) P2RX7MAOBMBOAT4SYKKMT2A
SCHEMBL2374158 0.80 KMT2A (0.46) P2RX7KMT2A
SCHEMBL8247000 0.79 ADORA2A (0.49) P2RX7ADORA2A
SCHEMBL15418113 0.79 MTNR1A (0.39) MBOAT4KMT2A
SCHEMBL29755971 0.78 P2RX7 (0.50) P2RX7MAOBADORA2AADAMTS4MMP13
SCHEMBL868879 0.78 P2RX7 (0.50) P2RX7MAOBADORA2AADAMTS4MMP13
SCHEMBL22396731 0.77 PSEN1 (0.42) P2RX7ADRB1HCRTR1HCRTR2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102917588-B Chemical compounds GLAXOSMITHKLINE LLC (US) 2014-10-08 CN disclosed
EP-2549868-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2013-01-30 EP disclosed
WO-2011119663-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed