SCHEMBL23742243

SCHEMBL23742243

CC(C)c1ccc(Cc2ccc(C#N)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.53
CYP2A6 P11509 2/20 0.52
SAE1 Q9UBE0 1/20 0.47
UBA2 Q9UBT2 1/20 0.47
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
CACNA1H O95180 1/20 0.43
IDO1 P14902 2/20 0.42
HRH3 Q9Y5N1 1/20 0.42
ALDH1A1 P00352 1/20 0.41
PANK3 Q9H999 2/20 0.41
ACACB O00763 1/20 0.41
IDH1 O75874 2/20 0.40
GRIA1 P42261 1/20 0.40
GRIA2 P42262 1/20 0.40
GRIA3 P42263 1/20 0.40
GRIA4 P48058 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
PYCR1 P32322 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL87339 0.87 CYP2A6 (0.52) LOXL2CYP2A6ALDH1A1PANK3GRIA1
SCHEMBL20373037 0.83 LOXL2 (0.44) LOXL2CYP2A6SAE1UBA2HRH3
SCHEMBL3956146 0.82 IDO1 (0.56) HTR1DHTR1BIDO1ALDH1A1PYCR1
SCHEMBL1344068 0.82 LOXL2 (0.65) LOXL2CYP2A6SAE1UBA2IDO1
SCHEMBL12263202 0.81 MMP3 (0.52) CYP2A6ALDH1A1PANK3GRIA1GRIA2
SCHEMBL27681566 0.80 LOXL2 (0.48) LOXL2CYP2A6SAE1UBA2IDO1
SCHEMBL1847770 0.79 LOXL2 (0.53) LOXL2CYP2A6CACNA1HALDH1A1PANK3
SCHEMBL31739252 0.77 MAOA (0.61) LOXL2CYP2A6SAE1UBA2HRH3
SCHEMBL14224119 0.77 CYP3A4 (0.64) LOXL2CYP2A6SAE1UBA2IDO1
SCHEMBL14346503 0.77 CYP2A6 (0.73) LOXL2CYP2A6SAE1UBA2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021156636-A1 TRIAZOLE DERIVATIVES WITH ANTIFUNGAL ACTIVITY KING'S COLLEGE LONDON (GB) 2021-08-12 WO disclosed