SCHEMBL23746997

SCHEMBL23746997

Cc1ccc2c(NS(=O)(=O)C3CCCC3)ncnn12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.43
KDR P35968 2/20 0.43
CHRNA7 P36544 1/20 0.41
HTR3A P46098 1/20 0.41
BRPF1 P55201 2/20 0.39
BRAF P15056 1/20 0.35
BRD4 O60885 4/20 0.34
EGLN2 Q96KS0 1/20 0.34
PIK3CA P42336 1/20 0.34
FPR1 P21462 2/20 0.33
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
CYP17A1 P05093 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GRM5 P41594 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23746999 0.99 EGFR (0.42) EGFRKDRCHRNA7HTR3ABRPF1
SCHEMBL23747016 0.85 CHRNA7 (0.41) CHRNA7HTR3ABRPF1BRAFBRD4
SCHEMBL23747109 0.84 CHRNA7 (0.41) CHRNA7HTR3ABRPF1BRAFBRD4
SCHEMBL23746995 0.78 FKBP1A (0.43) EGFRKDRCHRNA7HTR3AALDH1A1
SCHEMBL23746994 0.75 EGFR (0.45) EGFRKDRALDH1A1TSHR
SCHEMBL19864853 0.74 EGFR (0.55) EGFRKDRCHRNA7HTR3AALDH1A1
SCHEMBL23746986 0.74 EGFR (0.44) EGFRKDRCHRNA7HTR3ABRAF
SCHEMBL23747097 0.71 KDM4E (0.47) EGFRKDRALDH1A1
SCHEMBL23747000 0.70 EGFR (0.47) EGFRKDRPIK3CAALDH1A1TSHR
SCHEMBL23746992 0.70 EGFR (0.42) EGFRKDRCHRNA7HTR3ABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158516-A1 IRE1α MODULATORS AND USES THEREOF NIMBUS IASO, INC. (US) 2021-08-12 WO disclosed