SCHEMBL23747149

SCHEMBL23747149

O=S(=O)(CCC(F)(F)F)Nc1ncnn2c(Br)ccc12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CHRNA7 P36544 1/20 0.34
HTR3A P46098 1/20 0.34
KCNH2 Q12809 1/20 0.34
BRAF P15056 1/20 0.33
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23746992 0.85 EGFR (0.42) PTGS1PTGS2CHRNA7HTR3ABRAF
SCHEMBL23747216 0.84 EDNRB (0.40) CHRNA7HTR3AKCNH2BRAF
SCHEMBL23747204 0.74 AKR1B1 (0.37) CHRNA7HTR3AKCNH2
SCHEMBL23746985 0.73 ALDH1A1 (0.49) CHRNA7HTR3AKCNH2
SCHEMBL23747092 0.72 FFAR4 (0.44)
SCHEMBL23747015 0.72 CCR4 (0.42)
SCHEMBL23747030 0.71 FKBP1A (0.43) CHRNA7HTR3AKCNH2
SCHEMBL23747096 0.71 EDNRA (0.42)
SCHEMBL23747016 0.70 CHRNA7 (0.41) CHRNA7HTR3AKCNH2BRAF
SCHEMBL23746986 0.69 EGFR (0.44) PTGS1CHRNA7HTR3ABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158516-A1 IRE1α MODULATORS AND USES THEREOF NIMBUS IASO, INC. (US) 2021-08-12 WO disclosed