SCHEMBL23747756

SCHEMBL23747756

COc1ccc(CNC(=O)Nc2ccc(S(=O)(=O)c3ccccc3)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 16/20 0.77
NPC1 O15118 1/20 0.76
RAB9A P51151 1/20 0.76
SMN1; SMN2 Q16637 1/20 0.67
CYP2C9 P11712 2/20 0.63
HIF1A Q16665 1/20 0.62
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8175404 0.87 RAB9A (0.89) NAMPTNPC1RAB9ASMN1; SMN2HIF1A
SCHEMBL5427744 0.87 NPC1 (1.00) NPC1RAB9ASMN1; SMN2HIF1AHDAC1
SCHEMBL20379284 0.87 NAMPT (1.00) NAMPT
SCHEMBL17916794 0.85 SMN1; SMN2 (0.88) NAMPTNPC1RAB9ASMN1; SMN2HIF1A
SCHEMBL17831080 0.85 NPC1 (0.84) NAMPTNPC1RAB9ASMN1; SMN2HIF1A
SCHEMBL163178 0.83 NAMPT (1.00) NAMPTCYP2C9
SCHEMBL26101164 0.82 NPC1 (0.80) NAMPTNPC1RAB9ASMN1; SMN2HIF1A
SCHEMBL23747417 0.82 NPC1 (0.71) NAMPTNPC1RAB9ASMN1; SMN2HIF1A
SCHEMBL23747763 0.81 NPC1 (0.78) NPC1RAB9ASMN1; SMN2HIF1AHDAC1
SCHEMBL26097972 0.81 NPC1 (0.80) NPC1RAB9ASMN1; SMN2HIF1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
WO-2021159015-A1 NAMPT MODULATORS CYTOKINETICS, INC. (US) 2021-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 NAMPT 1/4885NPC1 463/4885RAB9A 807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.