SCHEMBL23749427

SCHEMBL23749427

CCOc1ccn(-c2ccccc2F)c(=O)c1C(=O)Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
AXL P30530 2/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 1/20 0.38
MET P08581 3/20 0.38
PLK4 O00444 1/20 0.38
ABL1 P00519 1/20 0.38
NTRK1 P04629 1/20 0.38
LCK P06239 1/20 0.38
RET P07949 1/20 0.38
KIT P10721 1/20 0.38
PDGFRA P16234 1/20 0.38
PRKACA P17612 1/20 0.38
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
ABL2 P42684 1/20 0.38
FRK P42685 1/20 0.38
MST1R Q04912 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15506051 0.89 L3MBTL1 (0.43) PTGS1PTGS2AXLMAPTTP53
SCHEMBL23749279 0.86 MET (0.42) AXLMAPTMETPLK4ABL1
SCHEMBL2592272 0.80 MET (0.51) AXLMAPTMETPLK4ABL1
SCHEMBL30031376 0.79 AXL (0.43) AXLKMT2AMETPLK4ABL1
SCHEMBL23749466 0.79 AXL (0.43) AXLKMT2AMETPLK4ABL1
SCHEMBL23749393 0.76 MET (0.43) AXLMAPTTP53KMT2AMET
SCHEMBL23749324 0.76 MET (0.41) AXLMAPTTP53METPLK4
SCHEMBL23770896 0.75 L3MBTL1 (0.43) AXLMAPTMETPLK4ABL1
SCHEMBL23749552 0.73 MAPK14 (0.54) MAPTTP53KMT2AALDH1A1POLB
SCHEMBL23749288 0.72 MAPK14 (0.48) MAPTTP53KMT2AL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220002308-A1 AROMATIC RING-LINKED DIOXINO-QUINAZOLINE OR DIOXINO-QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2022-01-06 US disclosed
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220002308-A1 AROMATIC RING-LINKED DIOXINO-QUINAZOLINE OR DIOXINO-QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF MERTK, AXL, TYRO3 PTGS1 3301/4885PTGS2 3905/4885AXL 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.