SCHEMBL23749451

SCHEMBL23749451

COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCCCC4)c4c(c23)OCCO4)c(F)c1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.64
AXL P30530 1/20 0.58
MST1R Q04912 1/20 0.58
TYRO3 Q06418 1/20 0.58
KIT P10721 2/20 0.57
KDR P35968 2/20 0.57
FLT3 P36888 2/20 0.57
PDGFRA P16234 1/20 0.57
RET P07949 1/20 0.55
PDGFRB P09619 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23749355 0.95 MET (0.64) METAXLMST1RTYRO3KIT
SCHEMBL23749544 0.94 MET (0.63) METAXLMST1RTYRO3KIT
SCHEMBL23749273 0.94 MET (0.64) METAXLMST1RTYRO3KIT
SCHEMBL23749503 0.91 MET (0.70) METAXLMST1RTYRO3KIT
SCHEMBL23749422 0.90 MET (0.76) METAXLMST1RTYRO3KIT
SCHEMBL23749511 0.90 MST1R (0.66) METAXLMST1RTYRO3KIT
SCHEMBL23749292 0.90 MET (0.63) METAXLMST1RTYRO3KIT
SCHEMBL23749432 0.89 MET (0.58) METAXLTYRO3KITKDR
SCHEMBL23749580 0.89 MET (0.62) METAXLMST1RTYRO3KIT
SCHEMBL23749520 0.88 MET (0.61) METAXLMST1RTYRO3KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed