SCHEMBL23749541

SCHEMBL23749541

O=C(Cl)c1cn(CCCN2CCOCC2)c(=O)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.43
MET P08581 3/20 0.43
AXL P30530 3/20 0.43
ATM Q13315 1/20 0.41
MAPK14 Q16539 3/20 0.40
CNR2 P34972 2/20 0.40
CNR1 P21554 1/20 0.40
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 2/20 0.40
MAPK13 O15264 2/20 0.40
MAPK12 P53778 2/20 0.40
MAPK11 Q15759 2/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
PCSK9 Q8NBP7 1/20 0.40
LMNA P02545 1/20 0.39
CD274 Q9NZQ7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969043 0.91 HTR3A (0.44) HTR3AMETAXLATMMAPK14
SCHEMBL30031006 0.90 PARP1 (0.44) HTR3AMETAXLATMMAPK14
SCHEMBL14967149 0.85 CNR1 (0.45) HTR3AMETAXLATMCNR2
SCHEMBL23749476 0.82 MET (0.47) METAXL
SCHEMBL23771043 0.80 MET (0.39) METAXLKDM4ELMNA
SCHEMBL23749310 0.80 AXL (0.41) METAXL
SCHEMBL22511523 0.76 AXL (0.52) METAXLCNR2CNR1
SCHEMBL23749414 0.76 MET (0.46) METAXL
SCHEMBL14966703 0.76 MET (0.48) HTR3AMETCNR2CNR1KDM4E
SCHEMBL23749366 0.76 MET (0.49) METAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12202835-B2 Substituted aromatic ring-linked dioxinoquinazolines and dioxinoquinolines as kinase inhibitors BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2025-01-21 US disclosed
CN-111196814-B Aromatic ring-linked dioxane quinazoline or quinoline compound, composition and application thereof 北京赛特明强医药科技有限公司 2022-12-06 CN disclosed
US-20220002308-A1 AROMATIC RING-LINKED DIOXINO-QUINAZOLINE OR DIOXINO-QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2022-01-06 US disclosed
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed
CN-111196814-A Aromatic ring connecting dioxane quinazoline or quinoline compound, composition and application thereof 北京赛特明强医药科技有限公司 2020-05-26 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220002308-A1 AROMATIC RING-LINKED DIOXINO-QUINAZOLINE OR DIOXINO-QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF MERTK, AXL, TYRO3 HTR3A 598/4885MET 14/4885AXL 2/4885
US-12202835-B2 Substituted aromatic ring-linked dioxinoquinazolines and dioxinoquinolines as kinase inhibitors MERTK, AXL, TYRO3 HTR3A 748/4885MET 12/4885AXL 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.