SCHEMBL30031006

SCHEMBL30031006

NC(=O)c1cn(CCCN2CCOCC2)c(=O)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.44
PARP2 Q9UGN5 2/20 0.44
HTR3A P46098 1/20 0.43
MET P08581 3/20 0.43
AXL P30530 3/20 0.43
MAPK14 Q16539 5/20 0.42
ATM Q13315 1/20 0.41
CNR2 P34972 2/20 0.40
CNR1 P21554 1/20 0.40
MAPK13 O15264 3/20 0.40
MAPK12 P53778 3/20 0.40
MAPK11 Q15759 3/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PCSK9 Q8NBP7 1/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969043 0.91 HTR3A (0.44) HTR3AMETAXLMAPK14ATM
SCHEMBL23749541 0.90 HTR3A (0.43) HTR3AMETAXLMAPK14ATM
SCHEMBL14967149 0.85 CNR1 (0.45) HTR3AMETAXLATMCNR2
SCHEMBL30031024 0.82 MET (0.47) METAXL
SCHEMBL14967452 0.82 MET (0.51) METAXLALDH1A1LMNA
SCHEMBL30031403 0.80 CA12 (0.39) METAXLKDM4ELMNA
SCHEMBL29814160 0.80 AXL (0.41) METAXL
SCHEMBL29814457 0.79 MET (0.45) METAXLLMNA
SCHEMBL29814274 0.78 MET (0.51) PARP1PARP2METAXL
SCHEMBL29626132 0.76 MET (0.46) METAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111196814-B Aromatic ring-linked dioxane quinazoline or quinoline compound, composition and application thereof 北京赛特明强医药科技有限公司 2022-12-06 CN disclosed