SCHEMBL2374960

SCHEMBL2374960

Cc1nc(C2CC2)ncc1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.51
KDM4E B2RXH2 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HTT P42858 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GABRP O00591 2/20 0.40
GABRD O14764 2/20 0.40
GABRA1 P14867 2/20 0.40
GABRB1 P18505 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40
GABRA5 P31644 2/20 0.40
GABRA3 P34903 2/20 0.40
GABRA2 P47869 2/20 0.40
GABRB2 P47870 2/20 0.40
GABRA4 P48169 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825471 0.85 NNMT (0.39) HPGDFOSJUNNFKB1NFKB2
SCHEMBL2374871 0.82 HPGD (0.37) HPGDKDM4ESMN1; SMN2ALDH1A1HTT
SCHEMBL3822431 0.81 POLB (0.37) HPGDKDM4EKMT2AMAPTSMN1; SMN2
SCHEMBL31324949 0.81 POLB (0.37) HPGDKDM4EKMT2AMAPTSMN1; SMN2
SCHEMBL27870383 0.79 GABRP (0.39) KDM4EKMT2AMAPTSMN1; SMN2ALDH1A1
SCHEMBL1014340 0.77 KDM4E (0.40) KDM4EKMT2ASMN1; SMN2HTTFOS
SCHEMBL21236319 0.75 FOS (0.32) HPGDFOSJUNNFKB1NFKB2
SCHEMBL10413068 0.74 PDE10A (0.36) KDM4EHTTFOSJUNNFKB1
SCHEMBL1434641 0.74 HPGD (0.61) HPGDKDM4EKMT2ASMN1; SMN2ALDH1A1
SCHEMBL19302651 0.74 PDE10A (0.39) KDM4EHTTFOSJUNNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2550264-B1 PYRIDAZINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2016-06-08 EP disclosed
US-9040537-B2 Pyridazine compounds for controlling invertebrate pests BASF SE (DE) 2015-05-26 US disclosed
EP-2550264-A1 PYRIDAZINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2013-01-30 EP disclosed
US-20130012380-A1 Pyridazine Compounds For Controlling Invertebrate Pests BASF SE (DE) 2013-01-10 US disclosed
WO-2011117286-A1 PYRIDAZINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2011-09-29 WO disclosed
EP-2019099-A1 Dpp-IV inhibitors Santhera Pharmaceuticals (Schweiz) AG (CH) 2009-01-28 EP disclosed
EP-2019099-A1 Dpp-IV inhibitors Santhera Pharmaceuticals (Schweiz) AG (CH) 2009-01-28 EP disclosed
WO-2009003681-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) AG (CH) 2009-01-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130012380-A1 Pyridazine Compounds For Controlling Invertebrate Pests GRIN2C, GRIN2A, NR2C2 HPGD 1662/4885KDM4E 2715/4885KMT2A 524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.