SCHEMBL23770872

SCHEMBL23770872

COc1ccc(NSc2cccc(N3CCCC(C)(C(=O)O)C3)n2)nc1-c1ccccc1C

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSA P10619 8/20 0.34
CYP1A2 P05177 3/20 0.33
CYP2C9 P11712 3/20 0.33
TSHR P16473 3/20 0.33
CYP2C19 P33261 3/20 0.33
HSD17B10 Q99714 3/20 0.33
CYP2D6 P10635 2/20 0.33
HPGD P15428 2/20 0.33
MAPK1 P28482 1/20 0.33
DGAT1 O75907 1/20 0.31
KCNH2 Q12809 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
ALDH1A1 P00352 2/20 0.30
CYP3A4 P08684 1/20 0.30
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770750 0.92 DGAT1 (0.32) CYP1A2CYP2C9TSHRCYP2C19HSD17B10
SCHEMBL23770738 0.90 SSTR5 (0.33) CYP1A2CYP2C9TSHRCYP2C19HSD17B10
SCHEMBL19970115 0.90 DGAT1 (0.34) DGAT1KCNH2HCRTR1HCRTR2CNR1
SCHEMBL23770774 0.88 PTGES (0.31) DGAT1KCNH2
SCHEMBL23770490 0.83 DGAT1 (0.30) DGAT1KCNH2
SCHEMBL19925808 0.83 CTSA (0.34) CTSACYP1A2CYP2C9TSHRCYP2C19
SCHEMBL19925805 0.83 CTSA (0.34) CTSACYP1A2CYP2C9TSHRCYP2C19
SCHEMBL29464511 0.83 CTSA (0.34) CTSACYP1A2CYP2C9TSHRCYP2C19
SCHEMBL19970116 0.83 DGAT1 (0.35) DGAT1KCNH2CNR1
SCHEMBL23770832 0.82 RBP4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed