SCHEMBL23774201

SCHEMBL23774201

CC1CNCc2ccc(OCc3ccccc3)cc21

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.54
HTR2C P28335 2/20 0.54
HRH3 Q9Y5N1 7/20 0.48
HTR2B P41595 1/20 0.47
MAOB P27338 4/20 0.45
MAOA P21397 3/20 0.45
ALOX5 P09917 1/20 0.44
CREBBP Q92793 1/20 0.44
CYP2D6 P10635 3/20 0.43
KDM1A O60341 1/20 0.43
HRH1 P35367 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5442266 0.88 HTR2C (0.65) HTR2AHTR2CHRH3HTR2BMAOB
SCHEMBL5442264 0.88 HTR2C (0.65) HTR2AHTR2CHRH3HTR2BMAOB
SCHEMBL5442260 0.88 HTR2C (0.65) HTR2AHTR2CHRH3HTR2BMAOB
SCHEMBL17583857 0.84 CA2 (0.46) HRH3MAOBMAOAALOX5CYP2D6
SCHEMBL4940018 0.82 HTR2C (0.67) HTR2AHTR2CHRH3HTR2BMAOB
SCHEMBL4940545 0.82 HTR2C (0.67) HTR2AHTR2CHRH3HTR2BMAOB
Hydrochloric Acid SCHEMBL4937772 0.81 HTR2C (0.66) HTR2AHTR2CHRH3HTR2BMAOB
Hydrochloric Acid SCHEMBL4929497 0.81 HTR2C (0.66) HTR2AHTR2CHRH3HTR2BMAOB
Hydrochloric Acid SCHEMBL4937777 0.81 HTR2C (0.66) HTR2AHTR2CHRH3HTR2BMAOB
SCHEMBL13198517 0.77 MAOA (0.53) HRH3MAOBMAOAALOX5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3194367-B1 TETRAHYDROISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR THE TREATMENT OF OBESITY AND DIABETES BOEHRINGER INGELHEIM INT (DE) 2021-08-18 EP disclosed