SCHEMBL23780360

SCHEMBL23780360

Cc1ccc(-c2ccc3nc(N)nc(NBr)c3c2)nc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.40
KCNH2 Q12809 2/20 0.39
ADORA2A P29274 2/20 0.38
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
APP P05067 3/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2A6 P11509 1/20 0.35
GRIA2 P42262 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
DHFR P00374 1/20 0.33
PDPK1 O15530 2/20 0.33
LCK P06239 1/20 0.33
KDR P35968 1/20 0.33
JAK3 P52333 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355092 0.89 HSP90AB1 (0.41) HSP90AB1KCNH2ADORA2ACCR1CCR5
SCHEMBL4364032 0.81 EGFR (0.55) KDR
SCHEMBL4358461 0.81 CD38 (0.43) CYP3A4PDPK1
SCHEMBL4364034 0.75 ADORA2A (0.40) HSP90AB1ADORA2ACCR1CCR5CCR8
SCHEMBL18041185 0.75 DHFR (0.53) KCNH2DHFR
SCHEMBL30943393 0.70 MAP4K4 (0.61)
SCHEMBL27960667 0.69 BACE1 (0.60) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL23780358 0.68 SRC (0.48) ADORA2ACYP3A4
SCHEMBL22745067 0.67 CCR1 (0.46) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL4351272 0.67 KCNH2 (0.43) HSP90AB1KCNH2ADORA2AAPPHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210276988-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. 2021-09-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210276988-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS NR3C1, NR3C2, NR4A1 HSP90AB1 4634/4885KCNH2 1412/4885ADORA2A 1163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.