SCHEMBL27960667

SCHEMBL27960667

Cc1ccc(-c2ccc3nc(N)ccc3c2)nc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 13/20 0.60
NCK1 P16333 1/20 0.60
CTSD P07339 1/20 0.52
PLAU P00749 1/20 0.46
NOS3 P29474 1/20 0.46
NOS2 P35228 1/20 0.46
CCR1 P32246 1/20 0.44
CCR5 P51681 1/20 0.44
CCR8 P51685 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NCF1 P14598 3/20 0.44
CYP3A4 P08684 1/20 0.41
CYP2A6 P11509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15344932 0.79 BACE1 (0.60) BACE1NCK1CTSDPLAUNOS3
SCHEMBL20929593 0.79 CCR1 (0.56) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL12386956 0.77 ALDH1A1 (0.62) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL7048523 0.76 BACE1 (1.00) BACE1NCK1CTSDPLAUNOS2
SCHEMBL31145084 0.76 CCR1 (0.52) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL13134511 0.76 CCR1 (0.52) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL4019673 0.75 NOS3 (0.69) NOS3NOS2CCR1CCR5CCR8
SCHEMBL5478956 0.74 BACE1 (0.62) BACE1NCK1CTSDPLAUNOS2
SCHEMBL27960721 0.74 BACE1 (0.57) BACE1NCK1CTSDPLAUNOS3
SCHEMBL29804792 0.74 PIK3CA (0.51) CCR1CCR5CCR8HDAC6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102574835-B Compounds for the treatment of cancer SPLICOS SOC 2014-04-16 CN claimed
CN-103948594-A Compounds for the treatment of cancer SPLICOS SOC 2014-07-30 CN disclosed
CN-102574835-B Compounds for the treatment of cancer SPLICOS SOC 2014-04-16 CN disclosed