SCHEMBL23794638

SCHEMBL23794638

CCOC(=O)c1sc(-c2cccc(Cl)c2)nc1C

nearest known ligand 0.80

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 5/20 0.80
KMT2A Q03164 2/20 0.70
CDC7 O00311 6/20 0.63
DBF4 Q9UBU7 6/20 0.63
MAPT P10636 5/20 0.63
KDM4E B2RXH2 3/20 0.63
ALDH1A1 P00352 3/20 0.63
LMNA P02545 1/20 0.56
MEN1 O00255 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.55
PDE4A P27815 1/20 0.51
PDE4B Q07343 1/20 0.51
PDE4C Q08493 1/20 0.51
PDE4D Q08499 1/20 0.51
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289979 0.90 TRPM8 (0.65) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL8867589 0.89 TRPM8 (1.00) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL12875919 0.87 CDC7 (0.66) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL28297244 0.87 CDC7 (0.65) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL299051 0.86 CDC7 (0.64) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL2881560 0.85 CDC7 (0.63) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL2885708 0.84 TRPM8 (0.78) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL1316281 0.84 CDC7 (0.77) TRPM8CDC7DBF4MAPTKDM4E
SCHEMBL3619382 0.84 CDC7 (0.62) TRPM8KMT2ACDC7DBF4MAPT
SCHEMBL8867138 0.84 CDC7 (0.62) TRPM8KMT2ACDC7DBF4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220009918-A1 Chemical Compounds GLAXOSMITHKLINE IP DEV LTD (GB) 2022-01-13 US disclosed
US-20220009918-A1 Chemical Compounds GLAXOSMITHKLINE IP DEV LTD (GB) 2022-01-13 US disclosed
EP-3877384-A1 CHEMICAL COMPOUNDS GlaxoSmithKline Intellectual Property Development Ltd (GB) 2021-09-15 EP disclosed
CN-112969698-A Chemical compound 葛兰素史密斯克莱知识产权发展有限公司 2021-06-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220009918-A1 Chemical Compounds HPGDS, PTGS1, PTGER1 TRPM8 3071/4885KMT2A 3678/4885CDC7 3467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.