SCHEMBL23833741

SCHEMBL23833741

COc1ccc([N+](=O)[O-])cc1S(=O)(=O)Nc1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.67
ALDH1A1 P00352 6/20 0.62
POLB P06746 3/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
ALPL P05186 6/20 0.61
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KMT2A Q03164 1/20 0.50
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25754684 0.87 HPGD (0.62) ALDH1A1POLBSMN1; SMN2ALPLLMNA
SCHEMBL25754679 0.86 SMN1; SMN2 (0.64) RECQLALDH1A1POLBSMN1; SMN2ALPL
SCHEMBL25754726 0.85 IDH1 (0.61) ALDH1A1POLBSMN1; SMN2ALPLLMNA
SCHEMBL23833756 0.85 POLB (0.56) ALDH1A1POLBSMN1; SMN2ALPLLMNA
SCHEMBL25754729 0.85 LMNA (0.67) RECQLALDH1A1POLBSMN1; SMN2ALPL
SCHEMBL25754730 0.84 MEN1 (0.61) RECQLALDH1A1POLBSMN1; SMN2ALPL
SCHEMBL25754693 0.84 POLB (0.55) ALDH1A1POLBSMN1; SMN2ALPLLMNA
SCHEMBL25754741 0.83 HPGD (0.57) ALDH1A1POLBALPLLMNAHPGD
SCHEMBL7527610 0.81 SMN1; SMN2 (0.65) ALDH1A1POLBSMN1; SMN2ALPLLMNA
SCHEMBL25754681 0.81 MEN1 (0.73) RECQLALDH1A1POLBSMN1; SMN2ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
EP-4121029-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF Amathus Therapeutics, Inc. (US) 2023-01-25 EP disclosed
WO-2021188880-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 RECQL 948/4885ALDH1A1 2569/4885POLB 1494/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.