SCHEMBL23846409

SCHEMBL23846409

O=C(Nc1cccc([S+]([O-])Nc2ccc(Br)cc2)c1)c1cnc(-c2ccccc2)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
MEN1 O00255 4/20 0.42
TP53 P04637 3/20 0.42
PIN1 Q13526 1/20 0.42
MMP2 P08253 3/20 0.40
MMP9 P14780 3/20 0.40
MMP8 P22894 3/20 0.40
MMP13 P45452 3/20 0.40
SENP1 Q9P0U3 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
LMNA P02545 1/20 0.38
ALOX15 P16050 1/20 0.38
COMT P21964 1/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25757044 0.78 MEN1 (0.53) KMT2AMEN1TP53ALDH1A1RAB9A
SCHEMBL3065306 0.74 NR1H4 (0.56) KMT2APIN1MMP2MMP9MMP8
SCHEMBL23833381 0.74 PIN1 (0.52) KMT2AMEN1TP53PIN1MMP2
SCHEMBL23840648 0.74 PIN1 (0.47) TP53PIN1MMP2MMP9MMP8
SCHEMBL25755108 0.73 RXFP1 (0.40) KMT2AMEN1RAB9ANPC1MAPK1
SCHEMBL23846523 0.73 RAB9A (0.41) KMT2AMEN1TP53ALDH1A1HPGD
SCHEMBL23846406 0.72 LMNA (0.47) KMT2AMEN1TP53PIN1ALDH1A1
SCHEMBL23846432 0.71 MAPT (0.45) KMT2AMEN1TP53PIN1ALDH1A1
SCHEMBL20841762 0.70 MAPT (0.60) KMT2AMEN1ALDH1A1HPGDNPC1
SCHEMBL4894537 0.70 MEN1 (0.49) KMT2AMEN1TP53PIN1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021188880-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed