SCHEMBL23848604

SCHEMBL23848604

O=S(=O)(Nc1cccc(C(F)(F)F)c1)N1CCOC(C(c2ccc(F)cc2)c2ccc(F)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.43
MAPT P10636 3/20 0.42
XBP1 P17861 1/20 0.42
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.40
MOGAT2 Q3SYC2 1/20 0.40
POLB P06746 1/20 0.39
SLC6A9 P48067 2/20 0.39
GRIN2B Q13224 1/20 0.39
MEN1 O00255 2/20 0.38
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP11B2 P19099 1/20 0.38
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
CHRM2 P08172 1/20 0.38
HTR1A P08908 1/20 0.38
DRD3 P35462 1/20 0.38
HTR2B P41595 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23832787 0.88 FKBP1A (0.43) TACR1MAPTMOGAT2POLBKMT2A
SCHEMBL23832785 0.87 KMT2A (0.42) MAPTHTTMOGAT2POLBSLC6A9
SCHEMBL30096698 0.87 KMT2A (0.42) MAPTHTTMOGAT2POLBSLC6A9
SCHEMBL25502088 0.86 KMT2A (0.40) MAPTHTTMOGAT2MEN1LMNA
SCHEMBL25501797 0.86 KMT2A (0.44) TACR1MOGAT2POLBMEN1KMT2A
SCHEMBL23848610 0.84 KMT2A (0.50) MOGAT2POLBMEN1KMT2AKDM4E
SCHEMBL25168299 0.82 FKBP1A (0.43) MAPTHTTMOGAT2POLBLMNA
SCHEMBL25501753 0.82 MAPT (0.46) TACR1MAPTXBP1HTTTSHR
SCHEMBL30096687 0.81 POLB (0.55) MAPTMOGAT2POLBKMT2A
SCHEMBL23832811 0.81 POLB (0.55) MAPTMOGAT2POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230146127-A1 3-DIARYLMETHYLENES AND USES THEREOF ATUX ISKAY LLC 2023-05-11 US disclosed
US-20230146127-A1 3-DIARYLMETHYLENES AND USES THEREOF ATUX ISKAY LLC 2023-05-11 US disclosed
WO-2021188949-A1 3-DIARYLMETHYLENES AND USES THEREOF ATUX ISKAY LLC (US) 2021-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230146127-A1 3-DIARYLMETHYLENES AND USES THEREOF MYC, MYCBP, FOXO1 TACR1 4866/4885MAPT 2576/4885XBP1 436/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.