Lysine

Lysine

SCHEMBL2385063

C[C@H](N)C(=O)O.C[C@H](N)C(=O)OC(=O)CN.NC(=O)CC[C@H](N)C(=O)OC[C@H](N)C(=O)O.NCC(=O)O.NCCCC[C@H](N)C(=O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.42
BLM P54132 2/20 0.40
ALOX15 P16050 1/20 0.40
PMP22 Q01453 1/20 0.40
KMT2A Q03164 1/20 0.40
NOD1 Q9Y239 1/20 0.32
CYP1A2 P05177 2/20 0.32
GRM8 O00222 1/20 0.32
GRM6 O15303 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIK1 P39086 1/20 0.32
GRM5 P41594 1/20 0.32
GRIA1 P42261 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA3 P42263 1/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
GRIA4 P48058 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530109 0.82 GSR (0.54) GSRBLMCYP1A2THRBNOS1
Lysine SCHEMBL8199478 0.80 GSR (0.65) GSRBLMCYP1A2GRM8GRM6
Alanine SCHEMBL4961214 0.80 GSR (0.59) GSRBLMCYP1A2THRBNOS1
Leucine SCHEMBL19692958 0.80 GSR (0.44) GSRGRIK1SLC1A3SLC1A2SLC1A1
Lysine SCHEMBL8885814 0.80 GSR (0.48) GSRBLMCYP1A2SLC1A3SLC1A2
SCHEMBL3650385 0.80 GSR (0.46) GSRBLMALOX15PMP22KMT2A
SCHEMBL233577 0.80 ALOX15 (0.44) GSRBLMALOX15PMP22KMT2A
Glutamine SCHEMBL8045598 0.79 GSR (0.67) GSRBLMALOX15PMP22KMT2A
Glutamine SCHEMBL19691979 0.79 GSR (0.67) GSRBLMALOX15PMP22KMT2A
Glutamine SCHEMBL2385066 0.78 GSR (0.54) GSRBLMALOX15PMP22KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8021646-B2 Compositions and methods for magnetic resonance imaging contrast agents NORTHWESTERN UNIVERSITY (US) 2011-09-20 US disclosed
US-20090053141-A1 COMPOSITIONS AND METHODS FOR MAGNETIC RESONANCE IMAGING CONTRAST AGENTS NORTHWESTERN UNIVERSITY (US) 2009-02-26 US disclosed
WO-2008073828-A2 COMPOSITIONS AND METHODS FOR MAGNETIC RESONANCE IMAGING CONTRAST AGENTS NORTHWESTERN UNIVERSITY (US) 2008-06-19 WO disclosed